Pentostatin is a purine antimetabolite and an adenosine deaminase (ADA) inhibitor (Ki = 0.09 nM).{23726,64635} It reduces 2'-deoxyadenosine-induced growth inhibition of MOLT-4 lymphoblast cells (Ki = 5.6 µM). It inhibits erythrocyte and ascites tumor ce
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A purine antimetabolite and an ADA inhibitor (Ki = 0.09 nM); reduces 2'-deoxyadenosine-induced growth inhibition of MOLT-4 lymphoblast cells (Ki = 5.6 µM); inhibits erythrocytes and ascites tumor cell ADA in an L1210 murine lymphocytic leukemia model at 0.2 mg/kg; inhibits tumor growth and increases survival rate in a CT26/NY-ESO-1 mouse xenograft model at 10 µg/mouse