URB602 is a selective inhibitor of monoacylglycerol lipase (MAGL), exhibiting an IC50 value of 28 µM for the rat brain enzyme.{13217} It does not inhibit fatty acid amide hydrolase (FAAH) at concentrations up to 100 µM or other lipid metabolizing enzyme
库存:
10 mg, 100 mg, 5 mg, 50 mg
供应商:
Cayman
CAS号:
565460-15-3
规格:
This biochemical is available in the following size(s) 25 mg, 5 mg, 50 mg - Please inquire
A selective inhibitor of MAGL (IC50 = 28 µM for the rat brain enzyme); does not inhibit FAAH at concentrations up to 100 µM or other lipid metabolizing enzymes such as diacylglycerol lipase or COX-2; inhibits glucose-stimulated and depolarization-induced insulin secretion in INS-1 cells