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Bafetinib
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Powder: -20°C, 3 years; 4°C, 2 years. In solvent: -80°C, 6 months; -20°C, 1 month.
INNO-406; NS-187
货期:1-2天
MedChemExpress LLC
10 mM * 1 mL/1 mg/5 mg/10 mg/50 mg/100 mg
MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
CAS No. : 859212-16-1
MCE 国际站:Bafetinib
产品活性:Bafetinib 是具有抗肿瘤活性的,有效的,具有口服活性的 Lyn/Bcr-Abl 酪氨酸激酶抑制剂。Bafetinib 通过 Bcl-2 家族调节的内在凋亡途径增强几种促凋亡的 Bcl-2 同源性 (BH) 3-纯蛋白 (Bim、Bad、Bmf 和 Bik) 的活性,并诱导 Ph+ 白血病细胞凋亡。
研究领域:Protein Tyrosine Kinase/RTK | Apoptosis
作用靶点:Bcr-Abl | Src | Apoptosis
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